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(αR,8aS)-GSK1614343 

Cat. No. M27777

All AbMole products are for research use only, cannot be used for human consumption.

(αR,8aS)-GSK1614343  Structure

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Quality Control & Documentation
Biological Activity

(αR,8aS)-GSK1614343 (compound 18a, d2) is a cyclized ghrelin antagonist with an pIC50 value of 8.4. (αR,8aS)-GSK1614343 shows a competitive antagonism of hGHSR1a with a mean pKb value of 8.06.

Chemical Information
Molecular Weight 487.44
Formula C22H23F6N5O
CAS Number 1092476-84-0
Form Solid
Storage Powder -20°C
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  Catalog
Abmole Inhibitor Catalog




Keywords: (αR,8aS)-GSK1614343  supplier, Ghrelin Receptor/GHSR, inhibitors, activators

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