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AF64394

Cat. No. M9494

All AbMole products are for research use only, cannot be used for human consumption.

AF64394 Structure
Synonym:

AF-64394

Size Price Availability Quantity
5mg USD 155 In stock
10mg USD 250 In stock
25mg USD 525 In stock
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Quality Control & Documentation
Biological Activity

AF64394 is a selective GPR3 inverse agonist with a pIC50 of 7.3.

Chemical Information
Molecular Weight 393.87
Formula C21H20ClN5O
CAS Number 1637300-25-4
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Jensen T, et al. Bioorg Med Chem Lett. The identification of GPR3 inverse agonist AF64394; the first small molecule inhibitor of GPR3 receptor function.

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  Catalog
Abmole Inhibitor Catalog




Keywords: AF64394, AF-64394 supplier, GPR/FFAR, inhibitors, activators

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