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Adrenorphin (Metorphamide) is a opioid octapeptide, acting as a potent agonist of μ-opioid receptor, with Ki of 12 nM. The binding ratios of Ki for μ-opioid receptor/Ki for δ-opioid receptor is 0.04, and the binding ratios of Ki for μ-opioid receptor/Ki for κ-opioid receptor is 0.46. Adrenorphin potently inhibits catecholamine secretion evoked by 10 μM nicotine in cultured human pheochromocytoma 6 cells, with IC50 of 1.1 μM.
| Molecular Weight | 984.18 |
| Formula | C44H69N15O9S |
| CAS Number | 88377-68-8 |
| Solubility (25°C) | DMSO 48 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[2] T Yanase, et al. J Clin Endocrinol Metab. Studies on adrenorphin in pheochromocytoma
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