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Adenosine receptor inhibitor 1

Cat. No. M40664

All AbMole products are for research use only, cannot be used for human consumption.

Adenosine receptor inhibitor 1 Structure

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Quality Control & Documentation
Biological Activity

Adenosine receptor inhibitor 1 is a potent, selective adenosine receptor inhibitor with Ki values of >1000, 68.5, >1000, >1000, >1000 nM for A1AR, A2AAR, A2BAR, and A3AR, respectively, and possesses analgesic as well as anti-inflammatory activity. It has analgesic and anti-inflammatory activities and can be used in cancer and neurodegenerative disease research.

Chemical Information
Molecular Weight 395.82
Formula C17H19ClFN5O3
CAS Number 2550400-52-5
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Anjali Saini et al. Eur J Med Chem. Adenosine receptor antagonists: Recent advances and therapeutic perspective

[2] Hillary A Johnston-Cox et al. J Cell Physiol. Physiological implications of adenosine receptor-mediated platelet aggregation

[3] Rosaria Volpini et al. Curr Pharm Des. Purine nucleosides bearing 1-alkynyl chains as adenosine receptor agonists

[4] P Narayan et al. Am J Physiol Heart Circ Physiol. Phosphatase inhibitor cantharidin blocks adenosine A(1) receptor anti-adrenergic effect in rat cardiac myocytes

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Keywords: Adenosine receptor inhibitor 1 supplier, Adenosine Receptor, inhibitors, activators

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