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Adenosine receptor antagonist 1

Cat. No. M40660

All AbMole products are for research use only, cannot be used for human consumption.

Adenosine receptor antagonist 1 Structure

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Biological Activity

Adenosine receptor antagonist 1 is a selective adenosine receptor A2aR antagonist with an IC50 value of 0.29 nM and a 14-fold higher selectivity for A2aR than for A2bR.

Chemical Information
Molecular Weight 447.85
Formula C22H15ClFN7O
CAS Number 2682930-40-9
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Catia Lambertucci et al. Curr Med Chem. A2A Adenosine Receptor Antagonists and their Potential in Neurological Disorders

[2] Anjali Saini et al. Eur J Med Chem. Adenosine receptor antagonists: Recent advances and therapeutic perspective

[3] Joana B Sousa et al. Recent Pat Anticancer Drug Discov. Adenosine Receptor Ligands on Cancer Therapy: A Review of Patent Literature

[4] A Nishiyama et al. J Pharmacol Exp Ther. Adenosine A(1) receptor antagonist KW-3902 prevents hypoxia-induced renal vasoconstriction

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Keywords: Adenosine receptor antagonist 1 supplier, Adenosine Receptor, inhibitors, activators

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