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4-Quinazolinamine

Cat. No. M3238

All AbMole products are for research use only, cannot be used for human consumption.

4-Quinazolinamine Structure
Synonym:

4-Aminoquinazoline, NSC 288012

Size Price Availability
100mg USD 180 Out of stock
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Quality Control & Documentation
Biological Activity

4-Quinazolinamine (4-Aminoquinazoline) is a potent and highly selective EGFR tyrosine kinase inhibitor. 4-Quinazolinamine (4-Aminoquinazoline) is useful as a fungicide and as an anti-inflammatory, antimicrobial and antihypertensive agent. Besides, the derivatives of 4-Quinazolinamine (4-Aminoquinazoline) is a novel class of opioid receptor like-1 (ORL1) antagonists.

Chemical Information
Molecular Weight 145.16
Formula C8H7N3
CAS Number 15018-66-3
Solubility (25°C) DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] No authors listed. Vandetanib

[2] No authors listed. Lapatinib

[3] No authors listed. Gefitinib

[4] Joseph W Polli, et al. The role of efflux and uptake transporters in [N-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamine (GW572016, lapatinib) disposition and drug interactions

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  Catalog
Abmole Inhibitor Catalog




Keywords: 4-Quinazolinamine, 4-Aminoquinazoline, NSC 288012 supplier, EGFR/HER2, inhibitors, activators

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