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(2S,3R)-LP99 is a potent and selective BRD7 and BRD9 inhibitor with an KD of 99 nM for BRD9. (2S,3R)-LP99 inhibits the association of BRD7 and BRD9 to acetylated histones in vitro and in cells. (2S,3R)-LP99 demonstrates that BRD7/9 plays a role in regulating pro-inflammatory cytokine secretion.
| Molecular Weight | 516.05 |
| Formula | C26H30ClN3O4S |
| CAS Number | 1808948-28-8 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
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