| Cat.No. | Name | Information |
|---|---|---|
| M6098 | Baicalein | Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor, IC50 value of 3.12 mM. |
| M9325 | EGTA | EGTA is a specific calcium chelator with a Kd of 60.5 nM at physiological pH (7.4) and a high specificity for Ca2+ than for Mg2+.EGTA significantly inhibits the substrate adhesion capacity of inflammatory macrophages. |
| M9330 | Brij-35 | Brij-35 (Polidocanol) is a high HLB, ethoxylated, nonionic ether of lauryl alcohol with broad pH stability. |
| M6154 | 2-PMPA tetrasodium | 2-PMPA (PMPA tetrasodium salt) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) with an IC50 of 300 pM. |
| M2250 | Pamidronate disodium | Pamidronate disodium is a nitrogen containing bisphosphonate, used to the research of preventing osteoporosis. |
| M9916 | DPPH | DPPH (2,2-Diphenyl-1-picrylhydrazyl) is a stable free radical that measures the free radical scavenging activity of antioxidants. |
| M9194 | Insulin (human) | Insulin (human) is a polypeptide hormone that regulates the level of sugar (glucose) in the blood and is produced by beta cells of islets. |
| M3409 | Formestane | Formestane is a second generation selective aromatase inhibitor with an IC50 of 80 nM. |
| M9665 | N-(2-amino-2-oxoethyl)acrylamide | N-(2-Amino-2-oxoethyl)acrylamide |
| M7791 | Exo-1 | Exo1 is a reversible inhibitor of exocytosis, also a Golgi ARF 1 (ADP-Ribosylation Factor) GTPase activator. |
| M10872 | Lufotrelvir | PF-07304814 IS A PHOSPHATE PRODRUG FOR PF-00835231 THAT BINDS AND INHIBITS SARS-CoV-2 3CLpro Active, Ki is 174 nM. |
| M10869 | OP-5244 | OP-5244 is a potent and orally active CD73 inhibitor,IC50 The value is 0.25 nM. OP-5244 reverses the immunosuppressive effect by blocking the production of adenosine, with the potential to conduct cancer research. |
| M10866 | NSC-70220 | NSC-70220 is a selective allosteric SOS1 inhibitor. NSC-70220 inhibits allosteric site activation and partially inhibits catalytic site activation. NSC-70220 has anti-cancer effects. |
| M10864 | Nicodicosapent | Nicodicosapent is a fatty acid niacin conjugate that inhibits the activity of sterol regulatory element binding proteins (SREBP) and the activity of proteins that regulate cholesterol metabolism such as PCSK9, HMG-CoA reductase, ATP citrate lyase, and NPC1L1. |
| M10863 | NCGC00378430 | NCGC00378430 is a potent inhibitor of the SIX1/EYA2 interaction. NCGC00378430 partially reverses SIX1 overexpression-mediated transcription and metabolic profiling, and reverses SIX1-induced TGF-β signaling and epithelial-interstitial transformation (EMT). NCGC00378430 inhibits SIX1-mediated breast cancer metastasis in mouse models. |
| M10851 | LY2922470 | LY2922470 is an effective, selective, orally potent GPR40 agonist that acts on human GPR40, mouse GPR40, and rat GPR40 EC50 The values are 7 nM, 1 nM, and 3 nM, respectively. LY2922470 lowers blood glucose levels while significantly increasing insulin and GLP-1, potentially for use in the study of type 2 diabetes mellitus (T2DM). |
| M10848 | LP-922761 | LP-922761 is a potent, selective, orally active AAK1 inhibitor in enzymatic and cell analysis IC50 4.8 nM and 7.6 nM, respectively. LP-922761 also inhibits BMP-2-induced protein kinase (BIKE),IC50 24 nM. LP-922761 has no significant activity against cell GAK, opioids, epinephrine alpha2, or GABAa receptors. |
| M10834 | Indeglitazar | Indeglitazar (PPM 204) is an orally active PPAR pan-agonist that acts on PPARα, PPARδ and PPARγ. |
| M10829 | HBF-0259 | HBF-0259 is a potent and selective hepatitis B virus (HBV) surface antigen (HBsAg) secretion inhibitor in HepG2.2.15 cells EC50 The value is 1.5 μM. HBF-0259 has no effect on HBV DNA synthesis. |
| M10825 | GSK-340 | |
| M10816 | FPTQ | FPTQ IS AN EFFECTIVE ONE mGluR1 antagonists, inhibiting people and rats IC50 The values are 6 nM and 1.4 nM, respectively. FPTQ has antioxidant and anti-inflammatory effects. |
| M10815 | Elobixibat | Elobixibat is a potent ileal bile acid transporter (IBAT) inhibitor, IC50 Values were 0.53±0.17 nM (human IBAT), 0.13±0.03 nM (mouse IBAT), 5.8± 1.6 nM (canine IBAT). |
| M10808 | CL264 | CL264 is a TLR7-specific agonist that can be used to study innate immune signaling pathways. |
| M10806 | CGX-1321 | |
| M10792 | BETd-246 | BETd-246 is a second-generation, PROTAC-based, BET bromine terminal domain (BRD) inhibitor that is connected by Cereblon ligands and BET ligands with good selectivity, efficacy and antitumor activity. |
| M10786 | Atuzaginstat | |
| M10778 | Aldumastat | Aldumastat (GLPG1972; S201086) is a potent, selective, orally active ADAMTS-5 (IC50=19 nM) inhibitor, whose selectivity is ADAMTS-4 (IC50=8 times 156 nM). Aldumastat has antimetabolic activity for osteoarthritis research. |
| M10769 | CS-2671 | TASP0415914 is an effective and orally active PI3Kγ inhibitor,IC50 29 nM. |
| M10768 | SKF83959 | SKF83959 is a potent selective dopamine D1-like Receptor partial agonist. SKF83959 Ki to rats D1，D5，D2AND D3 The values are 1.18, 7.56, 920, and 399 nM, respectively. SKF83959 is a potent sigma (σ)-1 receptor allosteric modulator. SKF83959 belongs to the benzazepine family and has an improving effect on cognitive dysfunction. SKF83959 can be used to study Alzheimer's disease and depression. |
| M10523 | L-Lysine hydrochloride | L-Lysine hydrochloride |
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