| Cat.No. | Name | Information |
|---|---|---|
| M1579 | Naloxone | Naloxone is an opioid inverse agonist used to counter the effects of opiate overdose. |
| M9615 | DAMGO | DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR. |
| M7014 | Naltrindole hydrochloride | Naltrindole hydrochloride is a selective non-peptide δ opioid antagonist (Ki = 0.02-0.3 nM), with much lower affinities for κ- and µ-opioid receptors (Kis = 10-66 and 6-64 nM, respectively). Naltrindole hydrochloride can cross the blood-brain barrier. |
| M52950 | Peptide E | Peptide E is a potent kappa opiate receptor agonist. |
| M52949 | Bilaid C | Bilaid C, a tetrapeptide, can be isolated from the Australian estuarine isolate of Penicillium sp. |
| M52948 | Dalargin | Dalargin is a potent δ-opioid receptor agonist. |
| M52947 | UFP-101 | UFP-101 is a potent, selective, and competitive antagonist of the NOP receptor, with a pKi of 10.24. |
| M52946 | ZP 120C | ZP 120C is a potent and partial ORL1 receptor agonist. |
| M52945 | CR 665 | CR 665 (JNJ 38488502) is a peripherally selective κ-opioid agonist. |
| M45206 | CVL-354 | CVL-354 is a potential best-in-class (BIC) kappa opioid receptor (KOR) antagonist for studies related to depression. |
| M45101 | Loxicodegol | Loxicodegol is a first-in-class, orally active, long-acting, selective μ-opioid agonist with structural properties that reduce its rate of crossing the blood-brain barrier compared to traditional μ-opioid agonists. |
| M41895 | Icalcaprant | Icalcaprant is a kappa-opioid receptor antagonist. |
| M41894 | MOR agonist-1 | MOR agonist-1 is a MOR (μ-opioid receptor) agonist. |
| M41893 | Deltorphin | Deltorphin (Deltorphin A; Dermenkephalin) is a biological active peptide. |
| M41892 | TIPP | TIPP is a potent and selective δ-opioid antagonist with a Ki value of 1.22 nM. |
| M41891 | DSLET | DSLET ([D-Ser2, Leu5, Thr6]-enkephalin) is a highly specific agonist of the δ-receptor. |
| M41890 | ICI 154129 | ICI 154 129 is a delta-opioid receptor antagonist and can be used for seizure research. |
| M41888 | BAN ORL 24 free base | BAN ORL 24 free base is a nociceptin/orphanin FQ (N/OFQ) peptide receptor (NOP) antagonist. |
| M41886 | MOR agonist-2 | MOR agonist-2 is a antagonist of D3R and agonist of MOR (Ki: 7.26 nM and 564 nM, respectively). |
| M41885 | GR 89696 free base | GR 89696 free base is a highly selective κ2 opioid receptor agonist with potential to prevent pruritus. |
| M41884 | SR16835 | SR16835 has high affinity for both NOPr and MOPr, with full agonist activity for NOPr and partial agonist activity for MOPr. |
| M38964 | Akuammidine | Akuammidine, isolated from the seeds of Picralima nitida, shows a preference for μ-opioid binding sites with Ki values of 0.6, 2.4 and 8.6 μM at μ-, σ- and κ-opioid binding sites, respectively. Akuammidine possesses anti-inflammatory and anti-asthmatic properties. |
| M31391 | TRV734 | TRV734 is an orally bioavailable G-protein-biased ligand for the μ-opioid receptor and an agonist for the μ-opioid receptor. |
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