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Opioid Receptor Opioid Receptor

Cat.No.  Name Information
M1579 Naloxone Naloxone is an opioid inverse agonist used to counter the effects of opiate overdose.
M9615 DAMGO DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR.
M7014 Naltrindole hydrochloride Naltrindole hydrochloride is a selective non-peptide δ opioid antagonist (Ki = 0.02-0.3 nM), with much lower affinities for κ- and µ-opioid receptors (Kis = 10-66 and 6-64 nM, respectively). Naltrindole hydrochloride can cross the blood-brain barrier.
M52993 Endomorphin 2 Endomorphin 2, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.
M52992 BAM-12P BAM-12P, an endogenous opioid peptide, is a novel pro-Met-enkephalin.
M52991 PL-017 PL-017 is a potent and selective μ opioid receptor agonist with an IC50 of 5.5 nM for 125I-FK 33,824 binding to μ site.
M52989 [Leu5]-Enkephalin, amide [Leu5]-Enkephalin, amide is a δ opioid receptor agonist.
M52987 Hemorphin-7 Hemorphin-7 is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.
M52986 [DPro10] Dynorphin A (1-11), porcine [DPro10] Dynorphin A (1-11), porcine, a N-Alkylated derivative, is a potent κ-opioid receptor agonist with a Ki value of 0.13 nM.
M52985 [DAla2] Dynorphin A (1-13), amide (porcine) [DAla2] Dynorphin A (1-13), amide (porcine) is a petide.
M52984 [DAla2, DArg6] Dynorphin A, (1-13) (porcine) [DAla2, DArg6] Dynorphin A, (1-13) (porcine) (DADAD) is an opioid peptide (dynorphinl-13, DYN) derivative found in porcine pituitary extracts.
M52983 (D-Met2, Pro5)-Enkephalinamide (D-Met2,Pro5)-Enkephalinamide is a highly potent opiate agonist, and shows antinociceptive activity.
M52982 [D-Ala2]-Met-Enkephalin [D-Ala2]-Met-Enkephalin, an opioid peptide, is a potent opioid agonist.
M52981 [D-Ala2]-Met-Enkephalinamide [D-Ala2]-Met-Enkephalinamide, an opioid peptide, is a potent opioid agonist.
M52980 [Met5]-Enkephalin, amide [Met5]-Enkephalin, amide is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.
M52979 [(pF)Phe4]Nociceptin(1-13)NH2 [(pF)Phe4]Nociceptin(1-13)NH2 is a highly potent and selective NOP receptor (OP4) agonist, with a pKi of 10.68 and a pEC50 of 9.31.
M52978 [Nphe1]Nociceptin(1-13)NH2 [Nphe1]Nociceptin(1-13)NH2, a novel nociceptin/orphanin FQ (NC) endogenous ligand, is a selective and competitive ociceptin receptor antagonist without any residual agonist activity.
M52977 [Arg14, Lys15]Nociceptin [Arg14,Lys15]Nociceptin is a highly potent and selective NOP receptor (ORL1; OP4) agonist, with an EC50 of 1 nM.
M52976 D-Ala-Gly-Phe-Met-NH2 monoacetate D-Ala-Gly-Phe-Met-NH2 monoacetate, an opioid peptide, is a potent opiate δ-receptor agonist.
M52975 β-Endorphin (1-27) (human) β-Endorphin (1-27) (human) is an opioid antagonist that binds μ-, δ-, and κ-opioid receptors with Kis of 5.31, 6.17, and 39.82 nM, respectively.
M52974 β-Endorphin (6-31), human β-Endorphin, an endogenous opioid neuropeptide, is an opioid receptor agonist.
M52973 2, 6-Dimethyl-L-tyrosine 2,6-Dimethyl-L-tyrosine (Dmt) is a tyrosine derivative that enhances receptor affinity, functional bioactivity and in vivo analgesia of opioid peptides.
M52972 Nociceptin (1-13), amide Nociceptin (1-13), amide is a potent ORL1 receptor (opioid receptor-like 1 receptor, OP4) agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain membranes.




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