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Opioid Receptor Opioid Receptor

Cat.No.  Name Information
M1579 Naloxone Naloxone is an opioid inverse agonist used to counter the effects of opiate overdose.
M9615 DAMGO DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR.
M7014 Naltrindole hydrochloride Naltrindole hydrochloride is a selective non-peptide δ opioid antagonist (Ki = 0.02-0.3 nM), with much lower affinities for κ- and µ-opioid receptors (Kis = 10-66 and 6-64 nM, respectively). Naltrindole hydrochloride can cross the blood-brain barrier.
M56291 LY2940094 tartrate LY2940094 (BTRX-246040) tartrate is a potent, brain penetrant, selective and orally available N/OFQ peptide (NOP) receptor antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM).
M56290 AR-M 1000390 hydrochloride  AR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2±0.9 nM for δ agonist potency.
M56289 (-)-U-50488 hydrochloride (-)-U-50488 hydrochloride ((-)-Trans-(1S,2S)-U-50488 hydrochloride) is a selective kappa-opioid receptor (KOR) agonist (b>Kd=2.2 nM) over μ-opioid receptor (MOR) (b>Kd=430 nM).
M54828 Tegileridine Tegileridine is the potent agonist of opioid receptor (MOR). Tegileridine is an oxa spiro derivative which reduces the side effects mediated by β-arrestin.
M54435 Morphiceptin Morphiceptin is a potent and specific agonist for morphine (μ) receptors.
M54425 [Met5]-Enkephalin, amide TFA [Met5]-Enkephalin, amide TFA is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.
M54363 DPDPE DPDPE, an opioid peptide, is a selective δ-opioid receptor (DOR) agonist with anticonvulsant effects.
M54289 Gluten Exorphin C Gluten exorphin C is an opioid peptide derived from wheat gluten.
M54280 N-terminally acetylated Leu-enkephalin N-terminally acetylated Leu-enkephalin is the N-terminally acetylated form of Leu-enkephalin.
M54236 [D-Ala2]leucine-enkephalin [D-Ala2]leucine-enkephalin, a delta opioid agonist, is a degradation resistant long-acting Leu-enkephalin.
M54139 Acetyl tetrapeptide-15 Acetyl tetrapeptide-15 is a synthetic peptide used in the cosmetics for sensitive skin.
M54134 Difelikefalin Difelikefalin (CR-845; FE-202845) is a peripherally restricted and selective agonist of kappa opioid receptor (KOR).
M53919 β-Casomorphin, bovine β-Casomorphin, bovine (β-Casomorphin-7 (bovine) ) is a opioid peptide with an IC50 of 14 μM in an Opioid receptors binding assay.
M53000 [DPen2, Pen5] Enkephalin [DPen2, Pen5] Enkephalin is a δ-opioid receptor selective analog of [Leu5]-Enkephalin.
M52999 (N-Me-Tyr1, N-Me-Arg7, D-Leu-NHEt8)-Dynorphin A (1-8) (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8) (E-2078), a stable Dynorphin A (1–8) analog, is a kappa opioid receptor (KOR) agonist.
M52998 β-Lipotropin (61-69) β-Lipotropin (61-69) is a potent opioid agonist.
M52997 β-Endorphin, equine β-Endorphin, equine is an endogenous opioid peptide, which binds at high affinity to both μ/δ opioid receptors.
M52996 Gluten Exorphin B5 Gluten Exorphin B5 is an exogenous opioid peptides derived from wheat gluten, acts on opioid receptor, increases postprandial plasma insulin level in rats.
M52995 Dermorphin Analog Dermorphin Analog is an analog of Dermorphin.
M52994 Dermorphin TFA Dermorphin TFA is a natural heptapeptide μ-opioid receptor (MOR) agonist found in amphibian skin.




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