| Cat.No. | Name | Information |
|---|---|---|
| M2347 | (+)-Bicuculline | (+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels. |
| M5442 | Baclofen | Baclofen is an orally active, selective metabotropic GABAB receptor (GABABR) agonist. Baclofen mimics the action of GABA and produces slow presynaptic inhibition through the GABAB receptor. Baclofen has high blood brain barrier penetrance. Baclofen has the potential for muscle spasticity research. |
| M5653 | Flumazenil | Flumazenil is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses. |
| M56475 | CI-966 hydrochloride | CI-966 hydrochloride is a potent, selective, orally active and brain-penetrant inhibitor of the GABA transporter GAT-1, with IC50s of 0.26 μM and 1.2 μM for hGAT-1, rGAT-1, respectively. |
| M56474 | CGP36216 hydrochloride | CGP36216 hydrochloride is a selective antagonist at GABA presynaptic receptor. |
| M56473 | SCH 50911 hydrochloride | SCH 50911 hydrochloride, (+)-(S)-5,5-dimethylmorpholinyl-2-acetic acid, a selective, orally-active and competitive γ-Aminobutyric acid B GABA(B) receptor antagonist, binds to GABA(B) receptor with IC50 of 1.1 μM. |
| M56472 | Lesogaberan napadisylate | Lesogaberan (AZD-3355) napadisylate is a potent and selective GABAB receptor agonist with an EC50 of 8.6 nM for human recombinant GABAB receptors. |
| M56471 | Lesogaberan hydrochloride | Lesogaberan (AZD-3355) hydrochloride is a potent and selective GABAB receptor agonist with an EC50 of 8.6 nM for human recombinant GABAB receptor. |
| M56470 | Loreclezole hydrochloride | Loreclezole hydrochloride, an antiepileptic compound, is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit containing receptors. |
| M56468 | Tetrahydrodeoxycorticosterone | Tetrahydrodeoxycorticosterone, an neurosteroid, is a potent positive allosteric modulator (PAM) of GABAA receptor. |
| M54859 | Alogabat | Alogabat (RG-7816) is a GABAA α5 receptor positive allosteric modulators (PAMs). |
| M52787 | CGP7930 | CGP7930 (3-(3’,5’-Di-tert-butyl-4’-hydroxy) phenyl-2, 2-dimethylpropanol) is a positive metabotropic GABAB receptor allosteric modulator. |
| M44709 | 3,4,5-Trimethoxy-trans-cinnamic acid | (E)-3,4,5-Trimethoxycinnamic acid (TMCA) is a cinnamic acid substituted by multi-methoxy groups. |
| M42191 | NCS-382 sodium | NCS-382 (sodium) is a potent GABA receptor antagonist. |
| M42190 | MRK-898 | MRK-898 is an orally active GABA(A) receptor modulator. |
| M42189 | ZAPA sulfate | ZAPA sulfate is an agonist at low affinity GABAA-receptors. |
| M42188 | Xilmenolone | Xilmenolone is a GABAA receptor positive allosteric modulator. |
| M42187 | NNC 05-2090 | NNC 05-2090 is a potent inhibitor of mGAT2, with a Ki of 1.4 μM. |
| M42186 | Arecaidine hydrobromide | Arecaidine hydrobromide, a pyridine alkaloid, is a potent GABA uptake inhibitor. |
| M42185 | Muscimol hydrochloride | Muscimol hydrochloride is a potent GABAA receptor agonist (EC50=0.2 μM), partial GABAC receptor agonist and inactive GABAB receptor agonist. |
| M42183 | Panadiplon | Panadiplon (FG 10571; PNU 78875), a benzodiazepine receptor, is a 5GABAA partial agonist. |
| M42182 | α5IA | α5IA (L-822179) is a selective α5 GABAA receptor inverse agonist with neuroprotective potential. |
| M42181 | 3-Methylglutaconic acid | 3-Methylglutaconic acid is the major metabolites accumulating in 3-Methylglutaconic aciduria (MGTA). |
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