| Cat.No. | Name | Information |
|---|---|---|
| M2347 | (+)-Bicuculline | (+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels. |
| M5442 | Baclofen | Baclofen is an orally active, selective metabotropic GABAB receptor (GABABR) agonist. Baclofen mimics the action of GABA and produces slow presynaptic inhibition through the GABAB receptor. Baclofen has high blood brain barrier penetrance. Baclofen has the potential for muscle spasticity research. |
| M5653 | Flumazenil | Flumazenil is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses. |
| M5870 | Pentylenetetrazol | Pentylenetetrazol displays activity as a central nervous system and respiratory stimulant. It is considered a non-competitive GABA(A) receptor antagonist. |
| M5730 | L-Cycloserine | L-cycloserine irreversibly inhibit GABA pyridoxal 5′-phosphate-dependent aminitransferase in E. coli, as well in the brains of various animals in a time-dependent manner, results in increased levels of gamma-aminobutyric acid (GABA), which is an inhibitory neurotransmitter in vivo. |
| M5669 | Gabapentin HCl | Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain. |
| M5575 | Dihydroergotoxine mesylate | Dihydroergotoxine mesylate is a complex of closely related alkaloid salts; Binds with high affinity to the GABAA receptor Cl- channel, producing an allosteric interaction with the benzodiazepine site. |
| M5390 | Afloqualone | Afloqualone is a agonist of GABA receptor . |
| M5378 | Acamprosate calcium | Acamprosate calcium (Campral EC) is a GABA receptor agonist and glutamate system modulator. |
| M5172 | 6-Prenylnaringenin | (2S)-6-Prenylnaringenin acts as a GABAA positive allosteric modulator at α+β- binding interface. |
| M4815 | Vigabatrin | Vigabatrin (γ-Vinyl-GABA), an inhibitory neurotransmitter GABA vinyl-derivative, is an orally active and irreversible GABA transaminase inhibitor. |
| M4441 | Jujuboside-A | Jujuboside A is A glycoside extracted from the Chinese traditional medicine ziziphus jujuboides, which can be used in studies on insomnia and anxiety symptoms. |
| M4231 | Ginkgolide-A | Ginkgolide A (BN-52020) is A GABA antagonist extracted from ginkgo biloba leaves. |
| M4073 | Ginsenoside-Rc | Ginsenoside Rc is one of the major ginsenosides. Ginsenoside Rc enhances GABA receptor A (GABAA) -mediated ion channel (IGABA) currents. Ginsenoside Rc also inhibited TNF-α and IL-1β expression. |
| M4019 | Songorine | Songorine is a diterpenoid alkaloid isolated from the genus Aconite. Songorine is a GABAA receptor antagonist in rat brain and has anticancer, anti-arrhythmia and anti-inflammatory activities. Songorine has potential to be used in epithelial ovarian cancer (EOC) studies. |
| M4013 | Glabridin | Glabridin, one of the active phytochemicals in licorice extract, binds to and activates the ligand binding domain of PPARγ, as well as the full length receptor. It is also a GABAA receptor positive modulator promoting fatty acid oxidation and improving learning and memory. |
| M3981 | Bilobalide | Bilobalide, a natural product extracted from Ginkgo biloba leaf, is known to exhibit a number of pharmacological activities. |
| M3968 | Dihydromyricetin | Dihydromyricetin is a natural antioxidant flavonoid from Ampelopsis grossedentata. |
| M3938 | Baicalin | Baicalin is an allosteric carnitine palmityl transferase 1 (CPT1) activator. Baicalin reduces the expression of NF-κB. |
| M3600 | Gabapentin | Gabapentin is a pharmaceutical agent, specifically a GABA analogue. |
| M3599 | Pregabalin | Pregabalin (Lyrica) is a 3-isobutyl derivative of gamma-amino butyric acid (GABA) with anti-convulsant, anti-epileptic, anxiolytic, and analgesic activities. |
| M3376 | Chlormezanone | Chlormezanone，a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm. |
| M3344 | Nefiracetam | Nefiracetam is a GABAergic, cholinergic, and monoaminergic neuronal systems enhancer for Ro 5-4864-induced convulsions. |
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