| Cat.No. | Name | Information |
|---|---|---|
| M3326 | Memantine hydrochloride | Memantine hydrochloride is a CYP2B6 and CYP2D6 inhibitor for recombinant CYP2B6 and CYP2D6 with Ki of 0.51 nM and 94.9 μM, respectively. |
| M2079 | Chrysin | Chrysin is a naturally occurring flavone chemically extracted from the passion flowers Passiflora caerulea. |
| M4000 | (±)-Naringenin | (±)-Naringenin, a common dietary flavonoid abundantly present in fruits and vegetables, is believed to possess strong anti-proliferative properties and the ability to induce apoptosis in hepatoma cell lines. |
| M14718 | Ipriflavone | Ipriflavone is a synthetic isoflavone derivative used to suppress bone resorption. |
| M14314 | N-Nornuciferine | N-Nornuciferine is an aporphine alkaloid in lotus leaf that significantly inhibits CYP2D6 with IC50 and Ki of 3.76 and 2.34 μM, respectively. |
| M14312 | Curcumenol | Curcumenol ((+)-Curcumenol) is a potent CYP3A4 inhibitor with an IC50 of 12.6 μM, which is one of constituents in the plants of medicinally important genus of Curcuma zedoaria, with neuroprotection, anti-inflammatory, anti-tumor and hepatoprotective activities. |
| M14311 | Cecropin B | Cecropin B has high level of antimicrobial activity and is considered as a valuable peptide antibiotic. |
| M14310 | Bergamottin | Bergamottin is a potent and competitive CYP1A1 inhibitor with a Ki of 10.703 nM. |
| M11528 | Naringin | Naringin, a flavanone glycoside, exerts various of pharmacological effects such as blood lipid lowering, antioxidant activity, anticancer activity, and inhibition of cytochrome P450 enzymes. |
| M11176 | Tebuconazole | Tebuconazole is an agricultural azole fungicide that also inhibits CYP51 for Candida albicans CYP51 (CaCYP51) and truncated human CYP51 (Δ60HsCYP51). IC50 The values are 0.9 and 1.3 μM, respectively. |
| M11164 | SDZ285428 | SDZ285428 is a CYP51 inhibitor. SDZ285428 suppresses Trypanosoma cruzi (TC) CYP51, I/E2 <1 (5 min) and I/E2=9 (1 h). SDZ285428 suppresses Trypanosoma brucei (TB) CYP51, I/E2 <1 (5 min) and I/E2=35 (1 h). |
| M11137 | Dihydromethysticin | Dihydroestherol (Dihydromethysticin) kava lactone, with induced CYP3A23 activity. |
| M10656 | Bergaptol | Bergaptol is a hydroxylated psoralen that acts as a potent inhibitors of debenzylation activity of CYP3A4 enzyme with an IC50 value of 24.92 uM. |
| M10488 | Phthalic acid mono-2-ethylhexyl ester (liquid) | Phthalic acid mono-2-ethylhexyl ester (MEHP) is a major bioactive metabolite of diethylhexyl phthalate (DEHP), which inhibits the 17, 20 lyase activity of CYP17. |
| M10057 | α-Naphthoflavone | α-Naphthoflavone is a potent and competitive aromatase inhibitor with an IC50 and a Ki of 0.5 and 0.2 μM, respectively. Alpha-Naphthoflavone can inhibit cell proliferation and induce apoptosis. |
| M9931 | ε-Viniferin | ε-Viniferin is a potent inhibitor for all the CYP family, with Ki values from 0.5-20 μM. |
| M9877 | Rhapontigenin | Rhapontigenin is a selective inactivator of cytochrome P450 1A1 with IC50 of 400 nM. |
| M9684 | (Rac)-Brassinazole | (Rac)-Brassinazole is a brassinosteroid (BR) biosynthesis inhibitor. |
| M9016 | Ezutromid | Ezutromid (BMN-195, SMT C1100) is a first-in-class oral bioavailable utrophin translational modulator with an EC50 value of 0.4 uM. |
| M8186 | Stiripentol | Stiripentol (BCX2600) can be used in the study of the third generation of antiepileptic drugs that enhance gaba energy neurotransmission. It's an inhibitor of cytochrome P450. |
| M7416 | TMS | TMS is a cytochrome P450 1B1 inhibitor. |
| M6451 | Apigenin | Apigenin is a competitive CYP2C9 inhibitor with a Ki of 2 μM. |
| M6389 | 1-Aminobenzotriazole (ABT) | 1-Aminobenzotriazole (ABT) is a cytochrome P450 inhibitor; inhibits 20-HETE synthesis. |
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