| Cat.No. | Name | Information |
|---|---|---|
| M2628 | Dexmedetomidine | Dexmedetomidine is a potent and highly selective α-2 adrenergic receptor agonist with sedative effects. |
| M3057 | Terbutaline Sulfate | Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM. |
| M3752 | Phentolamine Mesylate | Phentolamine mesylate is an orally active, rapid-acting alpha-adrenergic receptor antagonist, for the treatment of men suffering from erectile dysfunction (ED). |
| M2420 | Labetalol hydrochloride | Labetalol hydrochloride is a dual antagonist for both selective alpha1-adrenergic and nonselective beta-adrenergic receptors. |
| M13893 | Labetalol | Labetalol (AH5158) is an orally active selective α1- and non-selective β-adrenergic receptors competitive antagonist. |
| M5593 | Doxazosin Mesylate | Doxazosin, a quinazoline-derivative, selectively antagonizes postsynaptic α1-adrenergic receptors, used in the treatment of high blood pressure and urinary retention associated with benign prostatic hyperplasia. |
| M5462 | Bisoprolol fumarate | Bisoprolol fumarate is a selective type β1 adrenergic receptor blocker. |
| M7848 | ICI 118,551 hydrochloride | ICI 118,551 hydrochloride is a highly selective β2-adrenoceptor antagonist, with Kis of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively. |
| M2365 | Acebutolol hydrochloride | Acebutolol is a β-adrenergic receptors antagonist used in the treatment of hypertension, angina pectoris and cardiac arrhythmias. |
| M5784 | Metoprolol Succinate | Metoprolol Succinate (Toprol XL) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension. |
| M30268 | Cimaterol | Cimaterol (CL 263780) is a β-adrenergic agonist on energy metabolism in ob/ob mice. The Kd for Cimaterol binding to the L6 β-receptor is 26 nM which is compatible with its EC50 for the stimulation of protein synthesis (approx 5 nM). |
| M30248 | TD-5471 hydrochloride | TD-5471 hydrochloride is a potent and selective full agonist of the human β2-adrenoceptor. |
| M30236 | Alloyohimbine | Alloyohimbine, an alkaloid, is a selective α2-adrenoceptor antagonist with K Dα1, K Dα2 of 0.28 μM and 0.006 μM, respectively. |
| M30220 | Naphazoline nitrate | Naphazoline (Naphthazoline) nitrate is an α-adrenergic receptor agonist. Naphazoline nitrate reduces vascular hyperpermeability and promotes vasoconstriction. Naphazoline nitrate reduces the levels of inflammatory factors (TNF-α, IL-1β and IL-6), cytokines (IFN-γ and IL-4), IgE, GMCSF, and NGF。Naphazoline nitrate can be used for non-bacterial conjunctivitis research. |
| M30212 | Pronethalol hydrochloride | Pronethalol ((±)-Pronethalo) is a non-selective β-adrenergic antagonist. Pronethalol is a potent inhibitor of Sox2 expression. Pronethalol protects against and to reverse Digitalis-induced ventricular arrhythmias, and limits the cerebral arteriovenous malformation (AVMs). |
| M30198 | Mezilamine | Mezilamine is a potent antidopaminergic agent. Mezilamine induces a concentration dependent increase in the electrically stimulated overflow of 3H-noradrenaline from rat cortical slices, without affecting the basal overflow. Mezilamine acts as a presynaptic α-adrenoceptor antagonist and a postsynaptic α-adrenoceptor agonist. |
| M30002 | Zinterol | Zinterol (MJ 9184) is a potent and selective β2-adrenoceptor agonist. Zinterol increases ICa in a concentration-dependent manner with an EC50 of 2.2 nM. |
| M29947 | Levalbuterol | Levalbuterol ((R)-Albuterol; (R)-Salbutamol) is a short-acting β2-adrenergic receptor agonist and the active (R)-enantiomer of Salbutamol. Levalbuterol is a more potent bronchodilator than Salbutamol and has the potential for the treatment of COPD. |
| M29347 | N-5984 | N-5984 (KRP-204) is a potent and selective agonist of β3-adrenergic receptor. N-5984 has the potential for developing as one of the clinically effective drugs for obesity and diabetes mellitus. |
| M29250 | L-796568 | L-796568 is a β(3)-adrenergic receptor agonist. L-796568 can be used for the research of obesity. |
| M28518 | Carmoterol | Carmoterol is a highly potent, selective and long-acting β2-adrenoceptor agonist with the pEC50 of 10.19. Carmoterol has 53 times higher affinity for the β2-adrenoceptors than for the β1-adrenoceptors. Carmoterol can be used for the research of asthma and chronic obstructive pulmonary disease (COPD). |
| M28475 | Piribedil dihydrochloride | Piribedil dihydrochloride is a potent and orally active dopamine D2 and dopamine D3 agonist. Piribedil dihydrochloride is also a α2-adrenoceptors antagonist. Piribedil dihydrochloride can inhibit MLL1 methyltransferase activity (EC50: 0.18 μM). Piribedil dihydrochloride has the potential for the research of parkinson's disease, circulatory disorders, cancers. |
| M28242 | Piperoxan hydrochloride | Piperoxan (Benodaine) hydrochloride is an α2 adrenoceptor antagonist. Piperoxan hydrochloride is the first-generation antihistamine. |
| M28053 | Arformoterol maleate | Arformoterol ((R,R)-Formoterol) maleate, the (R,R)-enantiomer of Formoterol, is a long-acting β2-adrenergic receptor (β2-AR) agonist, with a Kd of 2.9 nM. Arformoterol maleate can be used for the research of chronic obstructive pulmonary disease (COPD). |
| M27928 | BI-167107 | BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM. |
| M27734 | Butyryltimolol | Butyryltimolol is the active precursor compound of Timolol, and is also a β-adrenergic (β-AR) blocker, which can pass through the cornea of the eye, and is enzymatically hydrolyzed to produce Timolol after entering the eye. |
| M25419 | A55453 | A55453 is a prazosin analogue and a potent α1-adrenergic antagonist. |
| M20992 | Bisoprolol | Bisoprolol is a cardioselective β1-adrenergic blocking agent used for secondary prevention of myocardial infarction (MI), heart failure, angina pectoris and mild to moderate hypertension. |
| M20963 | fluticasone furoate | Fluticasone furoate is an inhaled corticosteroid/long-acting beta-agonist combination with a prolonged bronchodilator duration of action. It is used for the treatment of non-allergic and allergic rhinitis administered by a nasal spray. |
| M20938 | Midodrine | Midodrine belongs to the class of medications known as vasopressors. It is an adrenergic alpha-1 agonist. |
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