| Cat.No. | Name | Information |
|---|---|---|
| M2628 | Dexmedetomidine | Dexmedetomidine is a potent and highly selective α-2 adrenergic receptor agonist with sedative effects. |
| M3057 | Terbutaline Sulfate | Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM. |
| M3752 | Phentolamine Mesylate | Phentolamine mesylate is an orally active, rapid-acting alpha-adrenergic receptor antagonist, for the treatment of men suffering from erectile dysfunction (ED). |
| M2420 | Labetalol hydrochloride | Labetalol hydrochloride is a dual antagonist for both selective alpha1-adrenergic and nonselective beta-adrenergic receptors. |
| M13893 | Labetalol | Labetalol (AH5158) is an orally active selective α1- and non-selective β-adrenergic receptors competitive antagonist. |
| M5593 | Doxazosin Mesylate | Doxazosin, a quinazoline-derivative, selectively antagonizes postsynaptic α1-adrenergic receptors, used in the treatment of high blood pressure and urinary retention associated with benign prostatic hyperplasia. |
| M5462 | Bisoprolol fumarate | Bisoprolol fumarate is a selective type β1 adrenergic receptor blocker. |
| M7848 | ICI 118,551 hydrochloride | ICI 118,551 hydrochloride is a highly selective β2-adrenoceptor antagonist, with Kis of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively. |
| M2365 | Acebutolol hydrochloride | Acebutolol is a β-adrenergic receptors antagonist used in the treatment of hypertension, angina pectoris and cardiac arrhythmias. |
| M5784 | Metoprolol Succinate | Metoprolol Succinate (Toprol XL) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension. |
| M41774 | Rezatomidine | Rezatomidine (AGN-203818) is a potent and selective α2-AR agonist. |
| M41773 | Xylometazoline | Xylometazoline is an α-adrenergic receptor agonist (Ki=0.05-1.7 μM). |
| M41772 | Bunazosin hydrochloride | Bunazosin hydrochloride is a potent and selective α1-adrenoceptor antagonist. |
| M41771 | Akuammigine | Akuammigine is an alkaloid that can be found in hook-bearing branch of Uncariarhynchophylla. |
| M41770 | Tiamenidine | Tiamenidine (HOE 440) is an orally active α2-adrenergic receptor agonist with antihypertensive effect. |
| M41769 | Bamosiran | Bamosiran is a small interfering RNA targeting β-adrenergic receptor 2, and is used to lower intraocular pressure |
| M41768 | Moprolol | Moprolol ((±)-Moprolol) is an beta-adrenergic receptor blocker, which can be used for research in essential hypertension. |
| M41767 | Norfenefrine hydrochloride | Norfenefrine hydrochloride is an orally active, endogenously found α-adrenergic agonist and can be used for the research of female stress incontinence. |
| M41766 | Benzquinamide hydrochloride | Benzquinamide (P2647) is an antiemetic which can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) with Ki values of 1,365, 691, and 545 nM, respectively. |
| M41765 | Spiroxatrine | Spiroxatrine (R 5188) is a selective, dual antagonist of 5-HT1α and α2-adrenergic, with the Ki values of 3.94, 224000, 118.5 nM for 5-HT1α, 5-HT1β and 5-HT2, respectively. |
| M41764 | Abediterol | Abediterol (LAS100977) is an inhaled long-acting β2-adrenoceptor agonist (LABA) and can be used for the research of asthma and chronic obstructive pulmonary disease (COPD). |
| M41635 | Etilefrine hydrochloride | Etilefrine hydrochloride is an orally active α adrenergic agonist. |
| M40941 | Guanadrel | Guanadrel is an orally active, spiroketal postganglionic adrenergic inhibitor containing a spirocyclic moiety in its structure, which may be used in studies related to hypertension. |
| M40721 | Mabuterol | Mabuterol is a selective, orally active beta-2 adrenergic receptor (β2-AR) agonist. Mabuterol inhibits PDGF-BB-induced cell proliferation, increased intracellular Ca2+, and Drp-1, cyclinD1, and PCNA protein expression, and enhances Mfn-2 expression. Can be used in studies of airway obstruction and chronic obstructive pulmonary disease (COPD). |
| M38956 | Dicentrine | Dicentrine is a natural product isolated from the plant Stephania epigaea Lo with antihypertensive effect. Dicentrine is an α1-adrenoceptor antagonist which has effective against human hyperplastic prostates. |
| M38955 | Terbutaline | Terbutaline is an orally active β2-adrenergic receptor agonist and an active metabolite of bambuterol. Terbutaline can be used in asthma symptom research. |
| M38954 | Clenbuterol | Clenbuterol (NAB-365) is a β2-adrenergic receptor agonist with an EC50 of 31.9 nM. Clenbuterol is a very potent inhibitor of the lipopolysaccharide (LPS)-induced release of TNF-α and IL-1β. Clenbuterol can inhibit the inflammatory process. Clenbuterol is a bronchodilator. |
| M31211 | ST91 | ST91 is a α2-adrenoceptor (α2AR) agonist. ST91 activates both α2AAR and non-α2AAR subtypes to produce spinal antinociception. |
| M31210 | Ractopamine | Ractopamine is a potent β-adrenergic receptor (βAR) agonist with Kd value of ~25 nM for pig β1AR and β2AR. Ractopamine is linked to protein metabolism. |
| M31209 | Hydroxybupropion | Hydroxybupropion is the major active metabolite of Bupropion. Hydroxybupropion inhibits norepinephrine uptake with an IC50 value of 1.7 μM. Hydroxybupropion is also a nACh receptor antagonist. |
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