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AChR/AChE Acetylcholine Receptors/Acetylcholinesterase

Cat.No.  Name Information
M2489 Carbachol chloride Carbachol is a cholinomimetic compound that binds and activates the acetylcholine receptor.
M3470 Oxybutynin Oxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties.
M3190 PNU-282987 PNU-282987 is a highly selective α7 nAChR agonist with Ki of 27 nM.
M5683 Glycopyrrolate Glycopyrrolate(Glycopyrronium Br) is a muscarinic competitive antagonist used as an antispasmodic.
M7227 EVP-6124 hydrochloride EVP-6124 hydrochloride) is a novel partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).
M8888 Donepezil Donepezil(E 2020) is a specific and potent AChE inhibitor for bAChE and hAChE with IC50 of 8.12 nM and 11.6 nM, respectively.
M5750 Lobeline HCl Lobeline hydrochloride, a nicotinic receptor agonist, acting as a potent antagonist at both α3β2 and α4β2 neuronal nicotinic receptor subtypes.
M3590 Butylscopolamine Bromide Butylscopolamine Bromide, is a peripherally acting antimuscarinic, anticholinergic agent used as an abdominal-specific antispasmodic.
M7940 Mecamylamine hydrochloride Noncompetitive nicotinic acetylcholine receptor antagonist; preferentially blocks nicotinic receptors at autonomic ganglia; crosses blood-brain barrier.
M30915 Pilocarpine  Pilocarpine is a selective M3-type muscarinic acetylcholine receptor (M3 muscarinic receptor) agonist.
M4590 Buddleoside Buddleoside
M4532 Rhodionin Rhodionin was isolated from the roots of Rhodiola crenulata and is a specific non-competitive cytochrome P450 2D6 inhibitor with IC50 of 0.761 μM and Ki of 0.769 μM. Rhodionin effectively inhibited acetylcholinesterase (AChE) in a dose-dependent manner with an IC50 range of 57.50 to 2.43 μg/mL. Rhodionin had effective DPPH radical scavenging activity with IC50 of 19.49 μM.
M4520 (+)-Corydaline Corydaline ((+) -corydaline) is an isoquinoline alkaloid extracted from Corydalis Yanhusuo. It is an inhibitor of AChE with IC50 of 226 µM. Corydaline is a μ-opioid receptor agonist (Ki = 1.23 µM) that inhibits the replication of enterovirus 71 (EV71) (IC50 = 25.23 µM). Corydaline has anti-angiogenesis, anti-allergy, gastric emptying and anti-nociception effects.
M4457 Jatrorrhizine chloride Jatrorrhizine chloride is a potent and orally active inhibitor of AChE (IC50=872 nM) over >115-fold selectivity for BuChE.
M4402 Epiberberine Epiberberine is a potent AChE and BChE inhibitor, and a non-competitive BACE1 inhibitor, with IC50s of 1.07, 6.03 and 8.55 μM, respectively. Epiberberine is also a potent inhibitor against both ureases with IC50 values of 3.0±0.01μM for HPU (ureases from Helicobacter pylori) and 2.3±0.01μM for JBU (ureases from jack bean).
M4391 Isoimperatorin Isoimperatorin is a methanol extract from the root of Angelica dahurica. It effectively inhibits acetylcholinesterase (AChE) with IC50 of 74.6 μM.
M4371 N-Methylcytisine N-methylcytisine (Caulophylline) is a tricyclic quinoline alkaloid with hypoglycemic, pain-relieving and anti-inflammatory activities. N-methylcytisine is a selective ligand of the acetylcholine acetylcholine receptor in the central nervous system and has a high affinity for the acetylcholine acetylcholine receptor in the optic ganglion of squid (Kd: 50 nM).
M4287 Picfeltarraenin-IB Picfeltarraenin IB is a triterpenoid compound that can be extracted from Picriafel-terrae Lour (P.fel-terrae). Picfeltarraenin IB is an inhibitor of acetylcholinesterase (AChE). Picfeltarraenin IB can be used to study infection, cancer and inflammation.
M4217 Timosaponin-A3 Timosaponin AIII could inhibit the activity of acetylcholinesterase (AChE) with IC50 value of 35.4 μM.
M4188 Tenuifolin Tenuifolin
M3893 TBPB TBPB is a novel highly selective agonist for the M(1) receptor with no agonist activity at any of the other mAChR subtypes.
M3650 Meclofenoxate hydrochloride Meclofenoxate hydrochloride is an ester of dimethylethanolamine (DMAE) and 4-chlorophenoxyacetic acid (pCPA).
M3606 Neostigmine Bromide Neostigmine Bromide is a reversible acetylcholinesterase inhibitor.
M3589 Methscopolamine bromide Methscopolamine is a muscarinic acetylcholine receptor blocker.
M3534 Pancuronium dibromide Pancuronium dibromide is a competitive acetylcholine antagonist with an IC50 of 5.5 nM.
M3530 Tolterodine tartrate Tolterodine tartrate is a tartrate salt of tolterodine that is a competitive muscarinic receptor antagonist.
M3501 Ipratropium Bromide Ipratropium Bromide is a muscarinic antagonist, bronchodilator, N-Isopropyl salt of atropine.
M3403 PNU-120596 PNU-120596 is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.
M3401 5-hydroxymethyl Tolterodine 5-hydroxymethyl tolterodine (PNU 200577) is a new muscarinic receptor antagonist with Kb of 0.84 nM.
M3393 Pyridostigmine Bromide Pyridostigmine Bromide is a parasympathomimetic and a reversible cholinesterase inhibitor.




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