| Cat.No. | Name | Information |
|---|---|---|
| M2147 | Ilomastat | Ilomastat (GM6001; Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor with Ki values of 0.4 nM, 0.5 nM, 27 nM, 3.7 nM, 0.1 nM, 0.2 nM, 3.6 nM, 13.4 nM and 0.36 nM for MMPs -1, -2, -3, -7, -8, -9, -12, -14 and -26, respectively. Ilomastat (GM6001; Galardin) reduces infarct volume following middle cerebral artery occlusion in an ischemic mouse model. |
| M4907 | Doxycycline Hyclate | Doxycycline is a member of the tetracycline antibiotics group, and is commonly used to treat a variety of infections. |
| M7413 | TMI 1 | TMI 1 is a adam 17 (TACE) and MMP inhibitor; orally bioavailable. |
| M9373 | T-5224 | T-5224 is a transcription factor c-Fos/activator protein (AP)-1 inhibitor with anti-inflammatory effects. |
| M4779 | Cordycepin | Cordycepin (3'-Deoxyadenosine) is a nucleoside derivative isolated from Cordyceps, inhibits IL-1β-induced MMP-1 and MMP-3 expression in rheumatoid arthritis synovial fibroblasts. |
| M11550 | 3-Aminopropionitrile fumarate | 3-amino-propanonitrile (β -amino-propanonitrile (BAPN)) acts as an irreversible inhibitor of lysyl oxidase (LOX), an enzyme involved in collagen cross-linking. |
| M11508 | Isoginkgetin | Isoginkgetin is a naturally occurring diflavone with antitumor activity. Isoginkgetin directly inhibits chymotrypsin-like, trypsin-like, and caspase - like activities of the 20S proteasome. Isoginkgetin is an inhibitor of MMP-9 and also an inhibitor of pre-mrna Splicing. |
| M9640 | MMP-9-IN-1 | MMP-9-IN-1 is a specific matrix metalloproteinase-9 (MMP-9) inhibitor. |
| M9466 | S-methyl-KE-298 | S-methyl-KE-298 is an active metabolite of KE-298. KE-298 inhibits matrix metalloproteinase (MMP-1) production from rheumatoid arthritis (RA) synovial cells. |
| M8732 | T-26c | T-26c is a highly potent, selective and cell-permeable matrix metalloproteinases 13 (MMP-13) inhibitor. |
| M8156 | SB-3CT | SB-3CT is a potent matrix metalloproteinase MMP-2 and MMP-9 inhibitor, with Ki values of 13.9 and 600 nM, respectively. SB-3CT shows blood-brain barrier permeability and has neuroprotective effects and anticancer activity. |
| M8041 | CP-101537 | Cp-101537 is an MMP inhibitor, a candidate compound for the treatment of myocardial infarction, and an antibacterial compound. |
| M7736 | CL-82198 | CL-82198 is a selective inhibitor of MMP-13 that displays no activity at MMP-1, MMP-9 or TACE. |
| M7454 | UK 356618 | UK 356618 is a potent and selective MMP-3 inhibitor. |
| M6749 | GI 254023X | GI 254023X is a selective ADAM10 metalloprotease inhibitor, with IC50 of 5.3 nM. |
| M6614 | CL 82198 hydrochloride | CL 82198 hydrochloride is a selective inhibitor of MMP-13. |
| M6463 | ARP 101 | ARP 101 is a selective inhibitor of MMP-2 that displays ~ 600-fold selectivity over MMP-1 (IC50 values are 0.81 and 486 nM respectively). |
| M6216 | TAPI-2 | TAPI-2 is a broad-spectrum inhibitor of matrix metalloprotease (MMP), tumour necrosis factorα-converting enzyme (TACE) and a disintegrin and metalloproteinase (ADAM), with an IC50 of 20±10 μM for MMP. |
| M6215 | TAPI-0 | TAPI-0 is an inhibitor which blocks the maturation of cytokines, soluble cyokine receptors and other proteins that require the action of proteases. |
| M4612 | Arctigenin | Arctigenin ((-) -arctigenin) is a bioactive lignan that can be used as an antitumor agent. Arctigenin has effective antioxidant, anti-inflammatory and antiviral activities. Arctigenin can be used to study metabolic disorders and central nervous system dysfunction. |
| M4473 | Morroniside | Morroniside plays a neuroprotective role by inhibiting neuronal apoptosis and mMP9/2 expression. |
| M4463 | Abametapir | Abametapir (HA-44, BRN 0123183) is an inhibitor of metalloproteinases critical for louse survival and egg development. |
| M4314 | Lucidenic-acid-A | Lucideric acid A, A natural product isolated from Ganoderma lucidum, can inhibit THE activity of MMP-9 induced by PMA, and has an anti-invasion effect on liver cancer cells. |
| M4311 | Lucidenic-acid-C | Lucidenic acid C, a natural product isolated from Ganoderma lucidum, can inhibit THE activity of MMP-9 induced by PMA, and has an anti-invasion effect on liver cancer cells. |
| M4210 | EGC | EGC is a potent inhibitor of amyloidogenic cystatin I66Q amyloid fibril formation in vitro, can bind to unfolded native polypeptides and prevent conversion to amyloid fibrils. |
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